Assay
Ref.
Price ( $ )
non-peptide receptors &
& Adenosine
A1 (antagonist radioligand)
0002
61
/
well
A1
G127
63
/
well
A1
0294
2103
/
cpd
non-peptide receptors &
& Adrenergic
alpha2 (non-selective) (antagonist radioligand)
0011
29
/
well
alpha2 (non-selective)
0297
1461
/
cpd
alpha2A (antagonist radioligand)
0013
61
/
well
alpha2A (agonist radioligand)
1669
61
/
well
alpha 2A
G120
63
/
well
beta2
0299
1461
/
cpd
beta2 (agonist radioligand)
0020
61
/
well
non-peptide receptors &
& Dopamine
D2S (antagonist radioligand)
0046
61
/
well
D2S (agonist radioligand)
1322
61
/
well
D2L (antagonist radioligand)
1405
61
/
well
D2
0310
1284
/
cpd
D3 (antagonist radioligand)
0048
61
/
well
D3 (agonist radioligand)
1660
61
/
well
D3
G016
63
/
well
non-peptide receptors &
& Glutamate
AMPA (agonist radioligand)
0064
40
/
well
NMDA (antagonist radioligand)
0066
40
/
well
PCP (antagonist radioligand)
0124
40
/
well
glycine (strychnine-insensitive) (antagonist radioligand)
0068
70
/
well
non-peptide receptors &
& Imidazoline
I2 (antagonist radioligand)
0081
40
/
well
non-peptide receptors &
& Muscarinic
M (non-selective) (antagonist radioligand)
0089
29
/
well
M1 (antagonist radioligand)
0091
61
/
well
M1
G029
63
/
well
M1
0318
1284
/
cpd
M2 (antagonist radioligand)
0093
61
/
well
M2 (agonist radioligand)
1626
61
/
well
M2
0319
2103
/
cpd
M3
G031
63
/
well
M3 (antagonist radioligand)
0095
61
/
well
M3
0320
1461
/
cpd
M4 (antagonist radioligand)
0096
61
/
well
M4 (agonist radioligand)
1619
61
/
well
M4
G032
63
/
well
M4 (inverse agonist effect)
2412
178
/
well
non-peptide receptors &
& Nicotinic
N neuronal alpha4beta2 (agonist radioligand)
3029
48
/
well
N neuronal alpha7 (antagonist radioligand)
3010
48
/
well
non-peptide receptors &
& Serotonin
5-HT (non-selective) (agonist radioligand)
0129
40
/
well
5-HT1A (agonist radioligand)
0131
61
/
well
5-HT1A
G044
63
/
well
5-HT1B (antagonist radioligand)
0132
40
/
well
5-HT1B
G126
63
/
well
5-HT2A (antagonist radioligand)
0135
61
/
well
5-HT2A (agonist radioligand)
0471
61
/
well
5-HT2A
G181
63
/
well
5-HT2A
0334
1284
/
cpd
5-HT2B (antagonist radioligand)
1609
61
/
well
5-HT2B (agonist radioligand)
1333
61
/
well
5-HT2B
0333
1461
/
cpd
5-HT2C (antagonist radioligand)
0137
61
/
well
5-HT2C (agonist radioligand)
1003
61
/
well
5-HT2C
G184
63
/
well
5-HT3 (antagonist radioligand)
0411
61
/
well
5-HT3
0335
1461
/
cpd
5-HT4
0336
1461
/
cpd
peptide receptors &
& Angiotensin-II
AT1 (antagonist radioligand)
0024
61
/
well
AT1
0301
1284
/
cpd
AT1
G052
63
/
well
AT2 (agonist radioligand)
0026
61
/
well
peptide receptors &
& Cytokines
IL-1beta (agonist radioligand) - custom offer
0073
inquire
IL-6 (agonist radioligand) - custom offer
0075
inquire
TNF-alpha (agonist radioligand)
0076
61
/
well
peptide receptors &
& Galanin
galanin (non-selective) (agonist radioligand)
0061
108
/
well
peptide receptors &
& Growth factors
TGF-beta (agonist radioligand) - custom offer
0071
inquire
VEGF (agonist radioligand) - custom offer
0672
inquire
peptide receptors &
& Neurokinin
NK1 (agonist radioligand)
0100
61
/
well
NK1
G085
63
/
well
NK1
0624
1461
/
cpd
peptide receptors &
& Neuropeptide Y
Y (non-selective) (agonist radioligand)
0105
48
/
well
Y1
0324
1284
/
cpd
peptide receptors &
& Neurotensin
NT (non-selective) (agonist radioligand)
0465
64
/
well
NT (non-selective)
0327
1461
/
cpd
peptide receptors &
& Somatostatin
sst (non-selective) (agonist radioligand)
0149
48
/
well
peptide receptors &
& Thyrotropin releasing hormone
TRH1 (agonist radioligand)
1616
61
/
well
TRH1
G098
63
/
well
peptide receptors &
& Vasopressin
V1a (agonist radioligand)
0159
61
/
well
V1a
G104
63
/
well
V1a
0338
1284
/
cpd
nuclear receptors &
& Steroid nuclear receptors
ER (non-selective) (agonist radioligand)
0152
70
/
well
ion channels &
& Intracellular ligand-gated channels
Ca2+ channels
IP3 (agonist radioligand)
0083
108
/
well
ion channels &
& Membrane ligand-gated channels
Glutamate
AMPA (agonist radioligand)
0064
40
/
well
NMDA (antagonist radioligand)
0066
40
/
well
PCP (antagonist radioligand)
0124
40
/
well
glycine (strychnine-insensitive) (antagonist radioligand)
0068
70
/
well
ion channels &
& Membrane ligand-gated channels
Nicotinic
N neuronal alpha4beta2 (agonist radioligand)
3029
48
/
well
N neuronal alpha7 (antagonist radioligand)
3010
48
/
well
ion channels &
& Membrane ligand-gated channels
Serotonin
5-HT3 (antagonist radioligand)
0411
61
/
well
5-HT3
0335
1461
/
cpd
ion channels &
& Voltage-gated channels
Ca2+ channels
L (dihydropyridine site) (antagonist radioligand)
0161
40
/
well
L (diltiazem site) (benzothiazepines) (antagonist radioligand)
0162
40
/
well
L (verapamil site) (phenylalkylamine) (antagonist radioligand)
0163
40
/
well
L
0339
1284
/
cpd
L (basal) - custom offer
0217
inquire
L (stimulated) - custom offer
0218
inquire
ion channels &
& Voltage-gated channels
K+ channels
KATP (antagonist radioligand)
0165
61
/
well
KATP
0340
1284
/
cpd
KV (antagonist radioligand)
0166
40
/
well
amine transporters &
& Choline
choline transporter (CHT1) (antagonist radioligand)
1552
61
/
well
choline transporter (antagonist radioligand) - custom offer
0098
inquire
amine transporters &
& Dopamine
dopamine transporter (antagonist radioligand)
0052
61
/
well
dopamine uptake
0394
64
/
well
amine transporters &
& Norepinephrine
norepinephrine transporter (antagonist radioligand)
0355
61
/
well
norepinephrine uptake
0393
64
/
well
amine transporters &
& Serotonin
5-HT transporter (antagonist radioligand)
0439
61
/
well
5-HT uptake
0392
61
/
well
Kinases &
& Protein-tyrosine kinases
RTK
VEGFR kinase
G142
44
/
cpd
VEGFR kinase (stimulant effect)
2696
26
/
well
VEGFR kinase (inhibitor effect)
2697
26
/
well
Kinases &
& Protein-tyrosine kinases
CTK
Tnk1
2785
19
/
well
Kinases &
& Protein-serine/threonine kinases
CMGC
CLK2
2019
19
/
well
ERK2 (P42mapk)
2878
13
/
well
GSK3alpha
2842
13
/
well
Kinases &
& Protein-serine/threonine kinases
CaMK
MARK1
3362
19
/
well
MARK2
1966
19
/
well
MARK3
2789
19
/
well
Kinases &
& Protein-serine/threonine kinases
AGC
GRK5
2020
19
/
well
PKCalpha
0348
13
/
well
PKCgamma
0350
19
/
well
Kinases &
& Protein-serine/threonine kinases
CK1
CK1alpha
1716
13
/
well
Non-kinase enzymes &
& Miscellaneous enzymes
xanthine oxidase/ superoxide O2- scavenging
0276
110
/
well
Non-kinase enzymes &
& NO synthases
constitutive NOS (cerebellar) - custom offer
0198
inquire
Non-kinase enzymes &
& Arachidonic acid metabolism
Phospholipase
sPLA2 (bee venom type III)
2999
110
/
well
sPLA2 (type V)
3176
141
/
well
Non-kinase enzymes &
& Arachidonic acid metabolism
Cyclooxygenases
COX2
0727
110
/
well
Non-kinase enzymes &
& Phosphatases
phosphatase PP1alpha
2656
110
/
well
phosphatase 2A (PP2A)
2584
110
/
well
Non-kinase enzymes &
& Monoamine & neurotransmitter synthesis & metabolism
acetylcholinesterase
0363
61
/
well
COMT (catechol-O-methyl transferase)
0457
70
/
well
MAO-A
0191
70
/
well
MAO-B
0621
70
/
well
tyrosine hydroxylase
0214
141
/
well
Non-kinase enzymes &
& Second messenger systems
Phospholipase C
PLC
2837
141
/
well
Non-kinase enzymes &
& Second messenger systems
Inositol phosphate
IP3 (agonist radioligand)
0083
108
/
well
Non-kinase enzymes &
& Proteases
Cysteine proteases
caspase-3
0774
141
/
well
caspase-6
0908
141
/
well
Non-kinase enzymes &
& Proteases
Aspartic proteases
BACE-1 (beta-secretase)
0701
141
/
well
cathepsin D
0650
141
/
well
cathepsin E
1001
141
/
well
Non-kinase enzymes &
& Proteases
Metalloproteases
ACE
0979
110
/
well
ACE
0302
1284
/
cpd
TACE
0702
110
/
well
specialized cellular assays &
& Monoamine & neurotransmitter release
dopamine release - custom offer
0450
inquire
norepinephrine release - custom offer
0460
inquire
5-HT release - custom offer
0459
inquire
specialized cellular assays &
& Cytokine secretion
IFN-gamma secretion - custom offer
0368
inquire
TNF-alpha secretion - custom offer
0259
inquire
IL-1beta secretion - custom offer
0262
inquire
IL-6 secretion - custom offer
0269
inquire
specialized cellular assays &
& Free radical secretion
superoxide O2- secretion - custom offer
0275
inquire
H2O2 secretion - custom offer
0277
inquire
H2O2 scavenging - custom offer
0278
inquire