Assay
Ref.
Price ( $ )
GPCRs
Adenosine
A1
G127
inquire
A1 (agonist effect)
2814
inquire
A1 (antagonist effect)
2820
inquire
A1 (inverse agonist effect)
2408
inquire
A2A
G002
inquire
A2A (agonist effect)
2055
inquire
A2A (antagonist effect)
2056
inquire
A2A (agonist effect)-custom offer
2527
inquire
A2A (inverse agonist effect)
2409
inquire
A2B
G003
inquire
A2B (agonist effect)
0452
inquire
A2B (antagonist effect)
0455
inquire
A3
G107
inquire
A3 (agonist effect)
0982
inquire
A3 (antagonist effect)
0983
inquire
GPCRs
Adrenergic
alpha1A
G004
inquire
alpha1A (agonist effect)
1500
inquire
alpha1A (antagonist effect)
1501
inquire
alpha1B
G005
inquire
alpha1B (agonist effect)
1901
inquire
alpha1B (antagonist effect)
1902
inquire
alpha2A
G120
inquire
alpha2A (agonist effect)
2558
inquire
alpha2A (antagonist effect)
2559
inquire
alpha2B
G011
inquire
alpha2B (agonist effect)
1813
inquire
alpha2B (antagonist effect)
1814
inquire
alpha2C
G006
inquire
alpha2C (agonist effect)
1736
inquire
alpha2C (antagonist effect)
1737
inquire
beta1
G007
inquire
beta1 (agonist effect)
1605
inquire
beta1 (antagonist effect)
1606
inquire
beta1 (inverse agonist effect)
2377
inquire
beta2
G008
inquire
beta2 (agonist effect)
1976
inquire
beta2 (antagonist effect)
1977
inquire
beta2 (inverse agonist effect)
2407
inquire
beta3
G009
inquire
beta3 (agonist effect)
2189
inquire
beta3 (antagonist effect)
2191
inquire
GPCRs
Angiotensin-II
AT1
G052
inquire
AT1 (agonist effect)
1912
inquire
AT1 (antagonist effect)
1913
inquire
GPCRs
Apelin
APJ (apelin)
G146
inquire
APJ (apelin) (agonist effect)
2844
inquire
APJ (apelin) (antagonist effect)
2850
inquire
GPCRs
Bombesin
BB1
G147
inquire
BB1 (agonist effect)
2846
inquire
BB1 (antagonist effect)
2852
inquire
BB2
G053
inquire
BB2 (agonist effect)
1915
inquire
BB2 (antagonist effect)
1916
inquire
BB3
G054
inquire
BB3 (agonist effect)
1319
inquire
BB3 (antagonist effect)
1764
inquire
GPCRs
Bradykinin
B1
G055
inquire
B1 (agonist effect)
1108
inquire
B1 (antagonist effect)
1109
inquire
B2
G056
inquire
B2 (agonist effect)
1263
inquire
B2 (antagonist effect)
1743
inquire
GPCRs
Calcitonin
CT (calcitonin)
G057
inquire
CT (calcitonin) (agonist effect)
1964
inquire
CT (calcitonin) (antagonist effect)
1965
inquire
GPCRs
Calcitonin gene-related peptide
CGRP
G058
inquire
CGRP (agonist effect)
1621
inquire
CGRP (antagonist effect)
1622
inquire
GPCRs
Calcium sensing
CaS
G010
inquire
CaS (agonist effect)
2144
inquire
CaS (antagonist effect)
2146
inquire
GPCRs
Cannabinoid
CB1
G012
inquire
CB1 (agonist effect)
1744
inquire
CB1 (antagonist effect)
1745
inquire
CB1 (inverse agonist effect)
2378
inquire
CB2
G013
inquire
CB2 (agonist effect)
1746
inquire
CB2 (antagonist effect)
1747
inquire
CB2 (inverse agonist effect)
2379
inquire
GPCRs
Chemokines
CCR2
G138
inquire
CCR2 (agonist effect)
2497
inquire
CCR2 (antagonist effect)
2501
inquire
CCR3
G148
inquire
CCR3 (agonist effect)
2136
inquire
CCR3 (antagonist effect)
2137
inquire
CXCR2 (IL-8B)
G113
inquire
CXCR2 (IL-8B) (agonist effect)
2480
inquire
CXCR2 (IL-8B) (antagonist effect)
2482
inquire
CXCR4
G114
inquire
CXCR4 (agonist effect)
2464
inquire
CXCR4 (antagonist effect)
2466
inquire
CCR1
G168
inquire
CCR1 (agonist effect)
2502
inquire
CCR1 (antagonist effect)
2503
inquire
GPCRs
Cholecystokinin
CCK1 (CCKA)
G062
inquire
CCK1 (CCKA) (agonist effect)
1876
inquire
CCK1 (CCKA) (antagonist effect)
1877
inquire
CCK2 (CCKB)
G063
inquire
CCK2 (CCKB) (agonist effect)
1878
inquire
CCK2 (CCKB) (antagonist effect)
1879
inquire
GPCRs
Complement 5a
C5a
G064
inquire
C5a (agonist effect)
2089
inquire
C5a (antagonist effect)
2098
inquire
GPCRs
Corticotropin releasing factor
CRF1
G065
inquire
CRF1 (agonist effect)
0504
inquire
CRF1 (antagonist effect)
0505
inquire
CRF2alpha
G066
inquire
CRF2alpha (agonist effect)
2085
inquire
CRF2alpha (antagonist effect)
2086
inquire
GPCRs
Dopamine
D1
G014
inquire
D1 (agonist effect)
1685
inquire
D1 (antagonist effect)
1686
inquire
D2S
G116
inquire
D2S (agonist effect)
2566
inquire
D2S (antagonist effect)
2569
inquire
D3
G016
inquire
D3 (agonist effect)
0683
inquire
D3 (antagonist effect)
0684
inquire
D4.4
G017
inquire
D4.4 (agonist effect)
1699
inquire
D4.4 (antagonist effect)
1700
inquire
D5
G018
inquire
D5 (agonist effect)
1688
inquire
D5 (antagonist effect)
1689
inquire
GPCRs
Endothelin
ETA
G067
inquire
ETA (agonist effect)
1264
inquire
ETA (antagonist effect)
2257
inquire
ETB
G068
inquire
ETB (agonist effect)
1762
inquire
ETB (antagonist effect)
1763
inquire
GPCRs
Free fatty acid
FFA1 (GPR40)
G123
inquire
FFA1 (GPR40) (agonist effect)
2665
inquire
FFA1 (GPR40) (antagonist effect)
2669
inquire
FFA2 (GPR43)
G132
inquire
FFA2 (GPR43) (agonist effect)
2710
inquire
FFA2 (GPR43) (antagonist effect)
2714
inquire
FFA3 (GPR41)
G143
inquire
FFA3 (GPR41) (agonist effect)
2819
inquire
FFA3 (GPR41) (antagonist effect)
2823
inquire
GPCRs
GABA
GABAB
G111
inquire
GABAB (agonist effect)
2525
inquire
GABAB (antagonist effect)
2526
inquire
GPCRs
Galanin
GAL2
G070
inquire
GAL2 (agonist effect)
1292
inquire
GAL2 (antagonist effect)
1893
inquire
GPCRs
Glucagon
GLP-1
G072
inquire
GLP-1 (agonist effect)
2181
inquire
GLP-1 (antagonist effect)
2182
inquire
secretin
G075
inquire
secretin (agonist effect)
2012
inquire
secretin (antagonist effect)
2014
inquire
GLP-2
G073
inquire
GLP-2 (agonist effect)
1993
inquire
GLP-2 (antagonist effect)
1998
inquire
glucagon
G074
inquire
glucagon (agonist effect)
1839
inquire
glucagon (antagonist effect)
1840
inquire
GPCRs
Glycoprotein hormone
TSH
G076
inquire
TSH (agonist effect)
2237
inquire
TSH (antagonist effect)
2239
inquire
GPCRs
Growth hormone-releasing hormone
GHRH
G071
inquire
GHRH (agonist effect)
2236
inquire
GHRH (antagonist effect)
2238
inquire
GPCRs
Histamine
H1
G115
inquire
H1 (agonist effect)
2542
inquire
H1 (antagonist effect)
2543
inquire
H2
G020
inquire
H2 (agonist effect)
1695
inquire
H2 (antagonist effect)
1696
inquire
H2 (inverse agonist effect)
2380
inquire
H3
G021
inquire
H3 (agonist effect)
1800
inquire
H3 (antagonist effect)
1801
inquire
H4
G125
inquire
H4 (agonist effect)
2595
inquire
H4 (antagonist effect)
2599
inquire
GPCRs
Leukotrienes
BLT1 (LTB4)
G023
inquire
BLT1 (LTB4) (agonist effect)
1245
inquire
BLT1 (LTB4) (antagonist effect)
1837
inquire
CysLT1 (LTD4)
G024
inquire
CysLT1 (LTD4) (agonist effect)
1383
inquire
CysLT1 (LTD4) (antagonist effect)
1607
inquire
CysLT2 (LTC4)
G025
inquire
CysLT2 (LTC4) (agonist effect)
2051
inquire
CysLT2 (LTC4) (antagonist effect)
2052
inquire
GPCRs
Lysophospholipid
Lysophosphatidic acid
LPA2
G144
inquire
LPA2 (agonist effect)
3171
inquire
LPA2 (antagonist effect)
3172
inquire
LPA3
G145
inquire
LPA3 (agonist effect)
3158
inquire
LPA3 (antagonist effect)
3170
inquire
GPCRs
Lysophospholipid
Sphingosine 1-phosphate
S1P1
G205
inquire
S1P1 (agonist effect)
3269
inquire
S1P1 (antagonist effect)
3271
inquire
S1P2
G026
inquire
S1P2 (agonist effect)
2133
inquire
S1P2 (antagonist effect)
2135
inquire
S1P3
G027
inquire
S1P3 (agonist effect)
2143
inquire
S1P3 (antagonist effect)
2145
inquire
GPCRs
Melanin concentrating hormone
MCH1
G077
inquire
MCH1 (agonist effect)
1035
inquire
MCH1 (antagonist effect)
1036
inquire
MCH2
G078
inquire
MCH2 (agonist effect)
1106
inquire
MCH2 (antagonist effect)
1107
inquire
GPCRs
Melanocortin
MC1
G079
inquire
MC1 (agonist effect)
2147
inquire
MC1 (antagonist effect)
2148
inquire
MC2
G080
inquire
MC2 (agonist effect)
2240
inquire
MC2 (antagonist effect)
2241
inquire
MC3
G081
inquire
MC3 (agonist effect)
0959
inquire
MC3 (antagonist effect)
1755
inquire
MC4
G082
inquire
MC4 (agonist effect)
0699
inquire
MC4 (antagonist effect)
0700
inquire
MC4 (inverse agonist effect)
2423
inquire
MC5
G083
inquire
MC5 (agonist effect)
1869
inquire
MC5 (antagonist effect)
1870
inquire
GPCRs
Melatonin
MT1 (ML1A)
G136
inquire
MT1 (ML1A) (agonist effect)
2498
inquire
MT1 (ML1A) (antagonist effect)
2500
inquire
MT2 (ML1B)
G028
inquire
MT2 (ML1B) (agonist effect)
2092
inquire
MT2 (ML1B) (antagonist effect)
2100
inquire
GPCRs
Motilin
motilin
G084
inquire
motilin (agonist effect)
1321
inquire
motilin (antagonist effect)
1894
inquire
GPCRs
Muscarinic
M1
G029
inquire
M1 (agonist effect)
1262
inquire
M1 (antagonist effect)
1474
inquire
M2
G030
inquire
M2 (agonist effect)
1658
inquire
M2 (antagonist effect)
1659
inquire
M2 (inverse agonist effect)
2411
inquire
M3
G031
inquire
M3 (agonist effect)
1243
inquire
M3 (antagonist effect)
1244
inquire
M4
G032
inquire
M4 (agonist effect)
1670
inquire
M4 (antagonist effect)
1671
inquire
M4 (inverse agonist effect)
2412
inquire
M5
G033
inquire
M5 (agonist effect)
1320
inquire
M5 (antagonist effect)
1652
inquire
GPCRs
Neurokinin
NK1
G085
inquire
NK1 (agonist effect)
2190
inquire
NK1 (antagonist effect)
2192
inquire
NK2
G086
inquire
NK2 (agonist effect)
1251
inquire
NK2 (antagonist effect)
1765
inquire
NK3
G087
inquire
NK3 (agonist effect)
1312
inquire
NK3 (antagonist effect)
1766
inquire
GPCRs
Neuromedin-U
NMU1
G194
inquire
NMU1 (agonist effect)
3310
inquire
NMU1 (antagonist effect)
3312
inquire
GPCRs
Neuropeptide S
NPS
G191
inquire
NPS (agonist effect)
3291
inquire
NPS (antagonist effect)
3292
inquire
GPCRs
Neuropeptide W / neuropeptide B
NPBW1
G171
inquire
NPBW1 (agonist effect)
2845
inquire
NPBW1 (antagonist effect)
2851
inquire
GPCRs
Neuropeptide Y
Y1
G088
inquire
Y1 (agonist effect)
2206
inquire
Y1 (antagonist effect)
2207
inquire
GPCRs
Neurotensin
NTS1 (NT1)
G089
inquire
NTS1 (NT1) (agonist effect)
1612
inquire
NTS1 (NT1) (antagonist effect)
1634
inquire
NTS2 (NT2)
G223
inquire
NTS2 (NT2) (agonist effect)
1919
inquire
NTS2 (antagonist effect)
1920
inquire
GPCRs
N-formyl peptide
fMLP
G069
inquire
fMLP (agonist effect)
2090
inquire
fMLP (antagonist effect)
2097
inquire
GPCRs
Opioid and opioid-like
delta2 (DOP)
G129
inquire
delta2 (DOP) (agonist effect)
2568
inquire
delta2 (DOP) (antagonist effect)
2571
inquire
kappa (KOP)
G090
inquire
kappa (KOP) (agonist effect)
2071
inquire
kappa (KOP) (antagonist effect)
2072
inquire
mu (MOP)
G091
inquire
mu (MOP) (agonist effect)
1392
inquire
mu (MOP) (antagonist effect)
1393
inquire
NOP (ORL1)
G119
inquire
NOP (ORL1) (agonist effect)
2381
inquire
NOP (ORL1) (antagonist effect)
2382
inquire
GPCRs
Orexin
OX1
G092
inquire
OX1 (agonist effect)
2234
inquire
OX1 (antagonist effect)
2235
inquire
OX2
G093
inquire
OX2 (agonist effect)
2349
inquire
OX2 (antagonist effect)
2350
inquire
GPCRs
Orphans (Class A)
GPR119
G189
inquire
GPR119 (agonist effect)
3297
inquire
GPR119 (antagonist effect)
3299
inquire
GPCRs
Parathyroid hormone
PTH1
G130
inquire
PTH1 (agonist effect)
2660
inquire
PTH1 (antagonist effect)
2661
inquire
GPCRs
Platelet activating factor
PAF
G034
inquire
PAF (agonist effect)
1610
inquire
PAF (antagonist effect)
1611
inquire
GPCRs
Prokineticin
PK1
G117
inquire
PK1 (agonist effect)
2449
inquire
PK1 (antagonist effect)
2451
inquire
PK2
G118
inquire
PK2 (agonist effect)
2450
inquire
PK2 (antagonist effect)
2452
inquire
GPCRs
Prostanoid
IP
G039
inquire
IP (agonist effect)
2228
inquire
IP (antagonist effect)
2229
inquire
DP1
G121
inquire
DP1 (agonist effect)
2484
inquire
DP1 (antagonist effect)
2486
inquire
EP1
G035
inquire
EP1 (agonist effect)
2053
inquire
EP1 (antagonist effect)
2054
inquire
EP2
G036
inquire
EP2 (agonist effect)
1956
inquire
EP2 (antagonist effect)
1957
inquire
EP3
G122
inquire
EP3 (agonist effect)
2577
inquire
EP3 (antagonist effect)
2578
inquire
EP4
G037
inquire
EP4 (agonist effect)
1871
inquire
EP4 (antagonist effect)
1872
inquire
FP
G038
inquire
FP (agonist effect)
2011
inquire
FP (antagonist effect)
2013
inquire
TP (TXA2/PGH2)
G040
inquire
TP (TXA2/PGH2) (agonist effect)
2059
inquire
TP (TXA2/PGH2) (antagonist effect)
2060
inquire
GPCRs
Proteinase-activated
PAR1
G109
inquire
PAR1 (agonist effect)
2332
inquire
PAR1 (antagonist effect)
2333
inquire
PAR2
G110
inquire
PAR2 (agonist effect)
2323
inquire
PAR2 (antagonist effect)
2324
inquire
GPCRs
Purinergic
P2Y1
G041
inquire
P2Y1 (agonist effect)
2132
inquire
P2Y1 (antagonist effect)
2134
inquire
P2Y2
G108