Assay
Ref.
Price ( $ )
Adenosine
adenosine transporter (antagonist radioligand)
0007
inquire
Cardiac toxicity
K+ channel
hERG
hERG (membrane preparation) (antagonist radioligand)
1868
inquire
Choline
choline transporter (CHT1) (antagonist radioligand)
1552
inquire
Dopamine
dopamine transporter (antagonist radioligand)
0052
inquire
dopamine transporter (antagonist radioligand) - custom offer
0051
inquire
GABA
GABA transporter (antagonist radioligand)
0060
inquire
GPCRs
Adenosine
A1 (antagonist radioligand)
0002
inquire
A1 (agonist radioligand)
0442
inquire
A1 (agonist radioligand) - custom offer
0001
inquire
A2A (agonist radioligand)
0004
inquire
A2B (antagonist radioligand)
0005
inquire
A3 (agonist radioligand)
0006
inquire
GPCRs
Adrenergic
alpha1 (non-selective) (antagonist radioligand)
0008
inquire
alpha1A (antagonist radioligand)
2338
inquire
alpha1A (antagonist radioligand)
0009
inquire
alpha1B (antagonist radioligand)
1633
inquire
alpha1B (antagonist radioligand) - custom offer
0010
inquire
alpha1D (antagonist radioligand)
1942
inquire
alpha2 (non-selective) (antagonist radioligand)
0011
inquire
alpha2A (antagonist radioligand)
0013
inquire
alpha2A (agonist radioligand)
3442
inquire
alpha2B (antagonist radioligand)
1344
inquire
alpha2B (antagonist radioligand) - custom offer
0014
inquire
alpha2C (antagonist radioligand)
0016
inquire
alpha2C (agonist radioligand)
3443
inquire
beta1 (agonist radioligand)
0018
inquire
beta1 (agonist radioligand) - custom offer
0017
inquire
beta2 (agonist radioligand)
0020
inquire
beta2 (agonist radioligand) - custom offer
0019
inquire
beta3 (antagonist radioligand)
0227
inquire
GPCRs
Angiotensin-II
AT1 (antagonist radioligand)
0024
inquire
AT2 (agonist radioligand)
0026
inquire
GPCRs
Apelin
APJ (apelin) (agonist radioligand)
2154
inquire
GPCRs
Bombesin
BB (non-selective) (agonist radioligand)
0030
inquire
BB1 (agonist radioligand)
2193
inquire
BB2 (agonist radioligand)
1986
inquire
BB3 (agonist radioligand)
0472
inquire
GPCRs
Bradykinin
B1 (agonist radioligand)
1189
inquire
B2 (agonist radioligand)
0033
inquire
GPCRs
Calcitonin
CT (calcitonin) (agonist radioligand)
0728
inquire
GPCRs
Calcitonin gene-related peptide
CGRP (agonist radioligand)
0373
inquire
GPCRs
Cannabinoid
CB1 (agonist radioligand)
0036
inquire
CB1 (agonist radioligand) - custom offer
0035
inquire
CB2 (agonist radioligand)
0037
inquire
GPCRs
Chemokines
CCR2 (agonist radioligand)
0362
inquire
CCR3 (agonist radioligand)
0481
inquire
CCR1 (agonist radioligand)
0361
inquire
CXCR2 (IL-8B) (agonist radioligand)
0419
inquire
CXCR4 (agonist radioligand)
1022
inquire
GPCRs
Cholecystokinin
CCK1 (CCKA) (agonist radioligand)
0039
inquire
CCK2 (CCKB) (agonist radioligand)
0041
inquire
GPCRs
Complement 5a
C5a (agonist radioligand)
0042
inquire
GPCRs
Corticotropin releasing factor
CRF1 (agonist radioligand)
1467
inquire
CRF2alpha (agonist radioligand)
2036
inquire
GPCRs
Dopamine
D1 (antagonist radioligand)
0044
inquire
D1 (antagonist radioligand) - custom offer
0043
inquire
D2S (antagonist radioligand)
0046
inquire
D2S (agonist radioligand)
1322
inquire
D2L (antagonist radioligand)
1405
inquire
D3 (antagonist radioligand)
0048
inquire
D3 (agonist radioligand)
1660
inquire
D4.4 (antagonist radioligand)
0049
inquire
D5 (antagonist radioligand)
0050
inquire
D5 (agonist radioligand)
1733
inquire
GPCRs
Endothelin
ETA (agonist radioligand)
0054
inquire
ETA (agonist radioligand) - custom offer
0053
inquire
ETB (agonist radioligand)
0056
inquire
ETB (agonist radioligand) - custom offer
0055
inquire
GPCRs
GABA
GABAB(1b) (antagonist radioligand)
0885
inquire
GABAB - custom offer
0059
inquire
GPCRs
Galanin
GAL1 (agonist radioligand)
0062
inquire
GAL2 (agonist radioligand)
0410
inquire
GPCRs
Glucagon
GLP-1 (agonist radioligand)
0228
inquire
glucagon (agonist radioligand)
1407
inquire
GPCRs
Gonadotrophin releasing hormone
GnRH (LH-RH) (agonist radioligand)
0456
inquire
GPCRs
Histamine
H1 (antagonist radioligand)
0870
inquire
H1 (antagonist radioligand)
0077
inquire
H2 (antagonist radioligand)
1208
inquire
H2 (antagonist radioligand)
0079
inquire
H3 (agonist radioligand)
1332
inquire
H3 (agonist radioligand)
0080
inquire
H4 (agonist radioligand)
1384
inquire
GPCRs
Leukotrienes
BLT1 (LTB4) (agonist radioligand)
1209
inquire
CysLT1 (LTD4) (agonist radioligand)
0086
inquire
CysLT2 (LTC4) (agonist radioligand)
2050
inquire
GPCRs
Lysophospholipid
Lysophosphatidic acid
LPA1 (agonist radioligand)
1468
inquire
GPCRs
Melanin concentrating hormone
MCH1 (agonist radioligand)
1115
inquire
MCH2 (agonist radioligand)
1190
inquire
GPCRs
Melanocortin
MC1 (agonist radioligand)
0644
inquire
MC3 (agonist radioligand)
0447
inquire
MC4 (agonist radioligand)
0420
inquire
MC5 (agonist radioligand)
0448
inquire
GPCRs
Melatonin
MT1 (ML1A) (agonist radioligand)
1538
inquire
MT2 (ML1B) (agonist radioligand)
1687
inquire
GPCRs
Motilin
motilin (agonist radioligand)
0470
inquire
GPCRs
Muscarinic
M (non-selective) (antagonist radioligand)
0089
inquire
M1 (antagonist radioligand)
0091
inquire
M1 (antagonist radioligand) - custom offer
0090
inquire
M2 (antagonist radioligand)
0093
inquire
M2 (agonist radioligand)
1626
inquire
M2 (antagonist radioligand) - custom offer
0092
inquire
M3 (antagonist radioligand)
0095
inquire
M4 (antagonist radioligand)
0096
inquire
M4 (agonist radioligand)
1619
inquire
M5 (antagonist radioligand)
0097
inquire
M5 (agonist radioligand)
1620
inquire
GPCRs
Neurokinin
NK1 (agonist radioligand)
0100
inquire
NK1 (agonist radioligand) - custom offer
0099
inquire
NK2 (agonist radioligand)
0102
inquire
NK3 (antagonist radioligand)
0104
inquire
NK3 (agonist radioligand)
1240
inquire
NK3 (agonist radioligand) - custom offer
0103
inquire
GPCRs
Neuromedin-U
NMU2 (agonist radioligand)
0991
inquire
GPCRs
Neuropeptide Y
Y (non-selective) (agonist radioligand)
0105
inquire
Y1 (agonist radioligand)
0106
inquire
Y2 (agonist radioligand)
0107
inquire
GPCRs
Neurotensin
NT (non-selective) (agonist radioligand)
0465
inquire
NTS1 (NT1) (agonist radioligand)
0109
inquire
GPCRs
N-formyl peptide
fMLP (agonist radioligand)
0407
inquire
GPCRs
Opioid and opioid-like
opioid (non-selective) (antagonist radioligand)
0112
inquire
delta2 (DOP) (agonist radioligand)
0114
inquire
kappa (KOP) (agonist radioligand)
1971
inquire
mu (MOP) (antagonist radioligand)
1666
inquire
mu (MOP) (agonist radioligand)
0118
inquire
mu (MOP) (agonist radioligand) - custom offer
0117
inquire
NOP (ORL1) (agonist radioligand)
0358
inquire
GPCRs
Orexin
OX1 (agonist radioligand)
1987
inquire
OX2 (agonist radioligand)
1988
inquire
GPCRs
Platelet activating factor
PAF (agonist radioligand)
0915
inquire
GPCRs
Prostanoid
IP (PGI2) (agonist radioligand)
2230
inquire
DP1 (agonist radioligand)
2517
inquire
EP1 (agonist radioligand)
0440
inquire
EP2 (agonist radioligand)
1955
inquire
EP3 (agonist radioligand)
2774
inquire
EP4 (agonist radioligand)
0441
inquire
FP (agonist radioligand)
1979
inquire
GPCRs
Proteinase-activated
PAR1 (agonist radioligand)
2592
inquire
PAR2 (agonist radioligand)
2424
inquire
GPCRs
Purinergic
P2Y (agonist radioligand)
0128
inquire
GPCRs
Relaxin
RXFP1 (agonist radioligand)
2058
inquire
GPCRs
Serotonin
5-HT (non-selective) (agonist radioligand)
0129
inquire
5-HT1A (agonist radioligand)
0131
inquire
5-HT1B (antagonist radioligand)
0132
inquire
5-HT1D (agonist radioligand)
1974
inquire
5-HT2A (antagonist radioligand)
0135
inquire
5-HT2A (agonist radioligand)
0471
inquire
5-HT2A (antagonist radioligand) - custom offer
0134
inquire
5-HT2B (antagonist radioligand)
1609
inquire
5-HT2B (agonist radioligand)
1333
inquire
5-HT2C (antagonist radioligand)
0137
inquire
5-HT2C (agonist radioligand)
1003
inquire
5-HT4e (antagonist radioligand)
0501
inquire
5-HT5a (agonist radioligand)
0140
inquire
5-HT6 (agonist radioligand)
0142
inquire
5-HT6 (agonist radioligand) - custom offer
0141
inquire
5-HT7 (agonist radioligand)
0144
inquire
5-HT7 (agonist radioligand) - custom offer
0143
inquire
GPCRs
Somatostatin
sst (non-selective) (agonist radioligand)
0149
inquire
sst1 (agonist radioligand)
1940
inquire
sst2 (agonist radioligand)
2339
inquire
sst4 (agonist radioligand)
0482
inquire
sst5 (agonist radioligand)
0626
inquire
GPCRs
Thyrotropin releasing hormone
TRH1 (agonist radioligand)
1616
inquire
GPCRs
Urotensin-II
UT (agonist radioligand)
1386
inquire
GPCRs
Vasoactive intestinal peptide
PAC1 (PACAP) (agonist radioligand)
1518
inquire
VPAC1 (VIP1) (agonist radioligand)
0157
inquire
VPAC2 (VIP2) (agonist radioligand)
0487
inquire
GPCRs
Vasopressin
V1a (agonist radioligand)
0159
inquire
V1a (agonist radioligand) - custom offer
0158
inquire
V1b (agonist radioligand)
0588
inquire
V1b (agonist radioligand) - custom offer
0466
inquire
V2 (agonist radioligand)
0497
inquire
V2 (agonist radioligand) - custom offer
0160
inquire
Intracellular ligand-gated channels
Ca2+ channels
IP3 (agonist radioligand)
0083
inquire
RY3 (ryanodine) (agonist radioligand)
0627
inquire
Membrane ligand-gated channels
GABA Channels
BZD (central) (agonist radioligand)
0028
inquire
Cl- channel (GABA-gated) (antagonist radioligand)
0170
inquire
GABAA1 (alpha 1,beta 2,gamma 2) (agonist radioligand)
3051
inquire
GABAA (agonist radioligand) - custom offer
0058
inquire
Membrane ligand-gated channels
Glutamate Channels
AMPA (agonist radioligand)
0064
inquire
kainate (agonist radioligand)
0065
inquire
NMDA (antagonist radioligand)
0066
inquire
PCP (antagonist radioligand)
0124
inquire
glycine (strychnine-insensitive) (antagonist radioligand)
0068
inquire
Membrane ligand-gated channels
Glycine Channels
glycine (strychnine-sensitive) (antagonist radioligand)
0067
inquire
Membrane ligand-gated channels
Nicotinic Channels
N muscle-type (antagonist radioligand)
0936
inquire
N muscle-type (antagonist radioligand) - custom offer
0111
inquire
N neuronal alpha4beta2 (agonist radioligand)
3029
inquire
N neuronal alpha4beta2 (agonist radioligand) - custom offer
0110
inquire
N neuronal alpha 7 (antagonist radioligand)
3010
inquire
Membrane ligand-gated channels
Purinergic Channels
P2X (agonist radioligand)
0127
inquire
Membrane ligand-gated channels
Serotonin Channels
5-HT3 (antagonist radioligand)
0411
inquire
Monoamine & neurotransmitter synthesis & metabolism
MAO-A (antagonist radioligand)
0443
inquire
Norepinephrine
norepinephrine transporter (antagonist radioligand)
0355
inquire
Nuclear receptors
Steroid nuclear receptors
AR (agonist radioligand)
0933
inquire
AR (agonist radioligand) - custom offer
0155
inquire
ER (non-selective) (agonist radioligand)
0152
inquire
ERalpha (agonist fluoligand)
0484
inquire
ERbeta (agonist fluoligand)
0485
inquire
PR (agonist radioligand)
2341
inquire
GR (agonist radioligand)
0469
inquire
Nuclear receptors
Non-steroid nuclear receptors
LXRbeta (agonist radioligand)
2047
inquire
PPARalpha (agonist radioligand)
0640
inquire
PPARgamma (agonist radioligand)
0641
inquire
PXR (agonist radioligand)
2538
inquire
RARalpha (agonist radioligand)
2084
inquire
TR (TH) (agonist radioligand)
0156
inquire
VDR (agonist radioligand)
0499
inquire
Other receptors
Atrial natriuretic peptide
ANP (agonist radioligand)
0027
inquire
Other receptors
Benzodiazepine
BZD (peripheral) (antagonist radioligand)
0029
inquire
Other receptors
Cytokines
TNF-alpha (agonist radioligand)
0076
inquire
IL-1beta (agonist radioligand) - custom offer
0073
inquire
IL-2 (agonist radioligand) - custom offer
0353
inquire
IL-4 (agonist radioligand) - custom offer
0074
inquire
IL-6 (agonist radioligand) - custom offer
0075
inquire
Other receptors
GABA
BZD (central) (agonist radioligand)
0028
inquire
Cl- channel (GABA-gated) (antagonist radioligand)
0170
inquire
GABA (non-selective) (agonist radioligand)
0057
inquire
GABAA1 (alpha 1,beta 2,gamma 2) (agonist radioligand)
3051
inquire
GABAA (agonist radioligand) - custom offer
0058
inquire
Other receptors
Glycine
glycine (strychnine-sensitive) (antagonist radioligand)
0067
inquire
Other receptors
Growth factors
EGF (agonist radioligand)
0069
inquire
PDGF (agonist radioligand)
0070
inquire
TGF-beta (agonist radioligand) - custom offer
0071
inquire
VEGF (agonist radioligand) - custom offer
0672
inquire
Other receptors
Imidazoline
I1 (agonist radioligand)
0642
inquire
I2 (antagonist radioligand)
0081
inquire
Other receptors
Insulin
insulin (agonist radioligand) - custom offer
0084
inquire
Other receptors
Melatonin
MT3 (ML2) (agonist radioligand)
0088
inquire
Other receptors
Nicotinic
N muscle-type (antagonist radioligand)
0936
inquire
N muscle-type (antagonist radioligand) - custom offer
0111
inquire
N neuronal alpha4beta2 (agonist radioligand)
3029
inquire
N neuronal alpha4beta2 (agonist radioligand) - custom offer
0110
inquire
N neuronal alpha 7 (antagonist radioligand)
3010
inquire
Other receptors
Purinergic
P2X (agonist radioligand)
0127
inquire
Other receptors
Serotonin
5-HT3 (antagonist radioligand)
0411
inquire
Other receptors
Sigma
sigma (non-selective) (agonist radioligand)
3500
inquire
sigma1 (agonist radioligand) - custom offer
0147
inquire
sigma1 (agonist radioligand)
0889
inquire
sigma2 (agonist radioligand)
3468
inquire
Phosphodiesterases
rolipram (antagonist radioligand)
0379
inquire
Serotonin
5-HT transporter (antagonist radioligand)
0439
inquire
5-HT transporter (antagonist radioligand) - custom offer
0145
inquire
Transduction signal enzymes
Inositol phosphate
IP3 (agonist radioligand)
0083
inquire
Voltage-gated channels
Ca2+ channels
Ca2+- L (dihydropyridine site) (antagonist radioligand)
0161
inquire
Ca2+- L (diltiazem site) (benzothiazepines) (antagonist radioligand)
0162
inquire
Ca2+- L (verapamil site) (phenylalkylamine) (antagonist radioligand)
0163
inquire
Ca2+- N (antagonist radioligand)
0164
inquire
Voltage-gated channels
K+ channels
hERG (membrane preparation) (antagonist radioligand)
1868
inquire
KATP (antagonist radioligand)
0165
inquire
KV (antagonist radioligand)
0166
inquire
SKCa (antagonist radioligand)
0167
inquire