Assay Ref. Price ( $ )
Adenosine
binding adenosine transporter (antagonist radioligand) 0007
inquire
Cardiac toxicity      K+ channel      hERG
binding hERG (membrane preparation) (antagonist radioligand) Human 1868
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Choline
binding choline transporter (CHT1) (antagonist radioligand) Human 1552
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Dopamine
binding dopamine transporter (antagonist radioligand) Human 0052
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binding dopamine transporter (antagonist radioligand) - custom offer 0051
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specific discount
GABA
binding GABA transporter (antagonist radioligand) 0060
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GPCRs      Adenosine
binding A1 (antagonist radioligand) Human 0002
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binding A1 (agonist radioligand) Human 0442
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binding A1 (agonist radioligand) - custom offer 0001
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specific discount
binding A2A (agonist radioligand) Human 0004
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binding A2B (antagonist radioligand) Human 0005
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binding A3 (agonist radioligand) Human 0006
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GPCRs      Adrenergic
binding alpha1 (non-selective) (antagonist radioligand) 0008
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binding alpha1A (antagonist radioligand) Human 2338
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binding alpha1A (antagonist radioligand) 0009
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binding alpha1B (antagonist radioligand) Human 1633
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binding alpha1B (antagonist radioligand) - custom offer 0010
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specific discount
binding alpha1D (antagonist radioligand) Human 1942
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binding alpha2 (non-selective) (antagonist radioligand) 0011
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binding alpha2A (antagonist radioligand) Human 0013
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binding alpha2A (agonist radioligand) Human 3442
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binding alpha2B (antagonist radioligand) Human 1344
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binding alpha2B (antagonist radioligand) - custom offer 0014
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specific discount
binding alpha2C (antagonist radioligand) Human 0016
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binding alpha2C (agonist radioligand) Human 3443
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binding new protocol beta1 (agonist radioligand) Human 0018
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binding beta1 (agonist radioligand) - custom offer 0017
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specific discount
binding beta2 (agonist radioligand) Human 0020
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binding beta2 (agonist radioligand) - custom offer 0019
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specific discount
binding beta3 (antagonist radioligand) Human 0227
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GPCRs      Angiotensin-II
binding AT1 (antagonist radioligand) Human 0024
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binding AT2 (agonist radioligand) Human 0026
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GPCRs      Apelin
binding APJ (apelin) (agonist radioligand) Human 2154
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GPCRs      Bombesin
binding BB (non-selective) (agonist radioligand) 0030
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binding BB1 (agonist radioligand) Human 2193
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binding BB2 (agonist radioligand) Human 1986
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binding BB3 (agonist radioligand) Human 0472
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GPCRs      Bradykinin
binding B1 (agonist radioligand) Human 1189
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binding B2 (agonist radioligand) Human 0033
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GPCRs      Calcitonin
binding CT (calcitonin) (agonist radioligand) Human 0728
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min 16 wells specific discount
GPCRs      Calcitonin gene-related peptide
binding CGRP (agonist radioligand) Human 0373
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GPCRs      Cannabinoid
binding CB1 (agonist radioligand) Human 0036
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binding CB1 (agonist radioligand) - custom offer 0035
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specific discount
binding CB2 (agonist radioligand) Human 0037
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GPCRs      Chemokines
binding CCR2 (agonist radioligand) Human 0362
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binding CCR3 (agonist radioligand) Human 0481
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min 16 wells
binding CCR1 (agonist radioligand) Human 0361
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binding CXCR2 (IL-8B) (agonist radioligand) Human 0419
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binding CXCR4 (agonist radioligand) Human 1022
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GPCRs      Cholecystokinin
binding CCK1 (CCKA) (agonist radioligand) Human 0039
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binding CCK2 (CCKB) (agonist radioligand) Human 0041
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GPCRs      Complement 5a
binding C5a (agonist radioligand) Human 0042
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min 16 wells specific discount
GPCRs      Corticotropin releasing factor
binding CRF1 (agonist radioligand) Human 1467
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binding CRF2alpha (agonist radioligand) Human 2036
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min 16 wells specific discount
GPCRs      Dopamine
binding D1 (antagonist radioligand) Human 0044
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binding D1 (antagonist radioligand) - custom offer 0043
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specific discount
binding D2S (antagonist radioligand) Human 0046
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binding D2S (agonist radioligand) Human 1322
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binding D2L (antagonist radioligand) Human 1405
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binding D3 (antagonist radioligand) Human 0048
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binding D3 (agonist radioligand) Human 1660
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binding D4.4 (antagonist radioligand) Human 0049
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binding D5 (antagonist radioligand) Human 0050
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binding D5 (agonist radioligand) Human 1733
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GPCRs      Endothelin
binding ETA (agonist radioligand) Human 0054
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binding ETA (agonist radioligand) - custom offer 0053
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specific discount
binding ETB (agonist radioligand) Human 0056
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binding ETB (agonist radioligand) - custom offer 0055
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specific discount
GPCRs      GABA
binding GABAB(1b) (antagonist radioligand) Human 0885
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binding GABAB - custom offer 0059
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GPCRs      Galanin
binding GAL1 (agonist radioligand) Human 0062
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binding GAL2 (agonist radioligand) Human 0410
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GPCRs      Glucagon
binding GLP-1 (agonist radioligand) 0228
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specific discount
binding glucagon (agonist radioligand) Human 1407
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GPCRs      Gonadotrophin releasing hormone
binding GnRH (LH-RH) (agonist radioligand) 0456
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min 16 wells specific discount
GPCRs      Histamine
binding H1 (antagonist radioligand) Human 0870
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binding H1 (antagonist radioligand) 0077
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specific discount
binding H2 (antagonist radioligand) Human 1208
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binding H2 (antagonist radioligand) 0079
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min 16 wells specific discount
binding H3 (agonist radioligand) Human 1332
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binding H3 (agonist radioligand) 0080
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binding H4 (agonist radioligand) Human 1384
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GPCRs      Leukotrienes
binding BLT1 (LTB4) (agonist radioligand) Human 1209
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binding CysLT1 (LTD4) (agonist radioligand) Human 0086
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binding CysLT2 (LTC4) (agonist radioligand) Human 2050
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specific discount
GPCRs      Lysophospholipid      Lysophosphatidic acid
binding LPA1 (agonist radioligand) Human 1468
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GPCRs      Melanin concentrating hormone
binding MCH1 (agonist radioligand) Human 1115
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binding MCH2 (agonist radioligand) Human 1190
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specific discount
GPCRs      Melanocortin
binding MC1 (agonist radioligand) 0644
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binding MC3 (agonist radioligand) Human 0447
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binding MC4 (agonist radioligand) Human 0420
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binding MC5 (agonist radioligand) Human 0448
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min 16 wells specific discount
GPCRs      Melatonin
binding MT1 (ML1A) (agonist radioligand) Human 1538
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binding MT2 (ML1B) (agonist radioligand) Human 1687
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GPCRs      Motilin
binding motilin (agonist radioligand) Human 0470
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GPCRs      Muscarinic
binding M (non-selective) (antagonist radioligand) 0089
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binding M1 (antagonist radioligand) Human 0091
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binding M1 (antagonist radioligand) - custom offer 0090
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specific discount
binding M2 (antagonist radioligand) Human 0093
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binding M2 (agonist radioligand) Human 1626
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binding M2 (antagonist radioligand) - custom offer 0092
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specific discount
binding M3 (antagonist radioligand) Human 0095
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binding M4 (antagonist radioligand) Human 0096
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binding M4 (agonist radioligand) Human 1619
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binding M5 (antagonist radioligand) Human 0097
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binding M5 (agonist radioligand) Human 1620
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GPCRs      Neurokinin
binding NK1 (agonist radioligand) Human 0100
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binding NK1 (agonist radioligand) - custom offer 0099
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specific discount
binding NK2 (agonist radioligand) Human 0102
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binding NK3 (antagonist radioligand) Human 0104
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binding NK3 (agonist radioligand) Human 1240
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binding NK3 (agonist radioligand) - custom offer 0103
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specific discount
GPCRs      Neuromedin-U
binding NMU2 (agonist radioligand) Human 0991
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GPCRs      Neuropeptide Y
binding Y (non-selective) (agonist radioligand) 0105
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binding Y1 (agonist radioligand) Human 0106
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binding Y2 (agonist radioligand) Human 0107
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GPCRs      Neurotensin
binding NT (non-selective) (agonist radioligand) 0465
inquire
min 16 wells specific discount
binding NTS1 (NT1) (agonist radioligand) Human 0109
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GPCRs      N-formyl peptide
binding fMLP (agonist radioligand) Human 0407
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min 16 wells specific discount
GPCRs      Opioid and opioid-like
binding opioid (non-selective) (antagonist radioligand) 0112
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binding delta2 (DOP) (agonist radioligand) Human 0114
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binding kappa (KOP) (agonist radioligand) 1971
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binding mu (MOP) (antagonist radioligand) Human 1666
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binding mu (MOP) (agonist radioligand) Human 0118
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binding mu (MOP) (agonist radioligand) - custom offer 0117
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specific discount
binding NOP (ORL1) (agonist radioligand) Human 0358
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GPCRs      Orexin
binding OX1 (agonist radioligand) Human 1987
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binding OX2 (agonist radioligand) Human 1988
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GPCRs      Platelet activating factor
binding PAF (agonist radioligand) Human 0915
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GPCRs      Prostanoid
binding IP (PGI2) (agonist radioligand) Human 2230
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binding DP1 (agonist radioligand) Human 2517
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binding EP1 (agonist radioligand) Human 0440
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binding EP2 (agonist radioligand) Human 1955
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binding EP3 (agonist radioligand) Human 2774
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specific discount
binding EP4 (agonist radioligand) Human 0441
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binding FP (agonist radioligand) Human 1979
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GPCRs      Proteinase-activated
binding PAR1 (agonist radioligand) Human 2592
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specific discount
binding PAR2 (agonist radioligand) Human 2424
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GPCRs      Purinergic
binding P2Y (agonist radioligand) 0128
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GPCRs      Relaxin
binding RXFP1 (agonist radioligand) Human 2058
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specific discount
GPCRs      Serotonin
binding 5-HT (non-selective) (agonist radioligand) 0129
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binding new protocol 5-HT1A (agonist radioligand) Human 0131
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binding 5-HT1B (antagonist radioligand) 0132
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binding 5-HT1D (agonist radioligand) 1974
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binding 5-HT2A (antagonist radioligand) Human 0135
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binding new protocol 5-HT2A (agonist radioligand) Human 0471
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binding 5-HT2A (antagonist radioligand) - custom offer 0134
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specific discount
binding 5-HT2B (antagonist radioligand) Human 1609
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binding 5-HT2B (agonist radioligand) Human 1333
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binding 5-HT2C (antagonist radioligand) Human 0137
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binding 5-HT2C (agonist radioligand) Human 1003
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binding 5-HT4e (antagonist radioligand) Human 0501
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binding 5-HT5a (agonist radioligand) Human 0140
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binding 5-HT6 (agonist radioligand) Human 0142
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binding 5-HT6 (agonist radioligand) - custom offer 0141
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specific discount
binding 5-HT7 (agonist radioligand) Human 0144
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binding 5-HT7 (agonist radioligand) - custom offer 0143
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specific discount
GPCRs      Somatostatin
binding sst (non-selective) (agonist radioligand) 0149
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binding sst1 (agonist radioligand) Human 1940
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binding sst2 (agonist radioligand) Human 2339
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min 16 wells specific discount
binding sst4 (agonist radioligand) Human 0482
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binding sst5 (agonist radioligand) Human 0626
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specific discount
GPCRs      Thyrotropin releasing hormone
binding TRH1 (agonist radioligand) Human 1616
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GPCRs      Urotensin-II
binding UT (agonist radioligand) Human 1386
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GPCRs      Vasoactive intestinal peptide
binding PAC1 (PACAP) (agonist radioligand) Human 1518
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binding VPAC1 (VIP1) (agonist radioligand) Human 0157
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binding new protocol VPAC2 (VIP2) (agonist radioligand) Human 0487
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GPCRs      Vasopressin
binding V1a (agonist radioligand) Human 0159
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binding V1a (agonist radioligand) - custom offer 0158
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specific discount
binding V1b (agonist radioligand) Human 0588
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binding V1b (agonist radioligand) - custom offer 0466
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specific discount
binding V2 (agonist radioligand) Human 0497
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binding V2 (agonist radioligand) - custom offer 0160
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specific discount
Intracellular ligand-gated channels      Ca2+ channels
binding IP3 (agonist radioligand) 0083
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min 16 wells specific discount
binding RY3 (ryanodine) (agonist radioligand) 0627
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min 16 wells specific discount
Membrane ligand-gated channels      GABA Channels
binding BZD (central) (agonist radioligand) 0028
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binding Cl- channel (GABA-gated) (antagonist radioligand) 0170
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binding GABAA1 (alpha 1,beta 2,gamma 2) (agonist radioligand) Human 3051
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binding GABAA (agonist radioligand) - custom offer 0058
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specific discount
Membrane ligand-gated channels      Glutamate Channels
binding AMPA (agonist radioligand) 0064
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binding new protocol kainate (agonist radioligand) 0065
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binding NMDA (antagonist radioligand) 0066
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binding PCP (antagonist radioligand) 0124
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binding glycine (strychnine-insensitive) (antagonist radioligand) 0068
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Membrane ligand-gated channels      Glycine Channels
binding new protocol glycine (strychnine-sensitive) (antagonist radioligand) 0067
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Membrane ligand-gated channels      Nicotinic Channels
binding new protocol N muscle-type (antagonist radioligand) Human 0936
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binding N muscle-type (antagonist radioligand) - custom offer 0111
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specific discount
binding N neuronal alpha4beta2 (agonist radioligand) Human 3029
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binding N neuronal alpha4beta2 (agonist radioligand) - custom offer 0110
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specific discount
binding new protocol N neuronal alpha 7 (antagonist radioligand) Human 3010
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Membrane ligand-gated channels      Purinergic Channels
binding P2X (agonist radioligand) 0127
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Membrane ligand-gated channels      Serotonin Channels
binding 5-HT3 (antagonist radioligand) Human 0411
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Monoamine & neurotransmitter synthesis & metabolism
binding MAO-A (antagonist radioligand) 0443
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Norepinephrine
binding norepinephrine transporter (antagonist radioligand) Human 0355
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Nuclear receptors      Steroid nuclear receptors
binding AR (agonist radioligand) Human 0933
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binding AR (agonist radioligand) - custom offer 0155
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specific discount
binding ER (non-selective) (agonist radioligand) Human 0152
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binding ERalpha (agonist fluoligand) Human 0484
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binding ERbeta (agonist fluoligand) Human 0485
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min 16 wells specific discount
binding PR (agonist radioligand) Human 2341
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binding GR (agonist radioligand) Human 0469
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Nuclear receptors      Non-steroid nuclear receptors
binding LXRbeta (agonist radioligand) Human 2047
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binding PPARalpha (agonist radioligand) Human 0640
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binding PPARgamma (agonist radioligand) Human 0641
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binding PXR (agonist radioligand) Human 2538
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binding RARalpha (agonist radioligand) Human 2084
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specific discount
binding TR (TH) (agonist radioligand) 0156
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binding VDR (agonist radioligand) Human 0499
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min 16 wells specific discount
Other receptors      Atrial natriuretic peptide
binding ANP (agonist radioligand) 0027
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min 16 wells specific discount
Other receptors      Benzodiazepine
binding BZD (peripheral) (antagonist radioligand) 0029
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Other receptors      Cytokines
binding TNF-alpha (agonist radioligand) Human 0076
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binding IL-1beta (agonist radioligand) - custom offer 0073
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specific discount
binding IL-2 (agonist radioligand) - custom offer 0353
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specific discount
binding IL-4 (agonist radioligand) - custom offer 0074
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specific discount
binding IL-6 (agonist radioligand) - custom offer Human 0075
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specific discount
Other receptors      GABA
binding BZD (central) (agonist radioligand) 0028
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binding Cl- channel (GABA-gated) (antagonist radioligand) 0170
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binding GABA (non-selective) (agonist radioligand) 0057
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binding GABAA1 (alpha 1,beta 2,gamma 2) (agonist radioligand) Human 3051
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binding GABAA (agonist radioligand) - custom offer 0058
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specific discount
Other receptors      Glycine
binding new protocol glycine (strychnine-sensitive) (antagonist radioligand) 0067
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Other receptors      Growth factors
binding EGF (agonist radioligand) Human 0069
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min 16 wells specific discount
binding PDGF (agonist radioligand) 0070
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binding TGF-beta (agonist radioligand) - custom offer 0071
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specific discount
binding VEGF (agonist radioligand) - custom offer Human 0672
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specific discount
Other receptors      Imidazoline
binding I1 (agonist radioligand) 0642
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binding new protocol I2 (antagonist radioligand) 0081
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Other receptors      Insulin
binding insulin (agonist radioligand) - custom offer 0084
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specific discount
Other receptors      Melatonin
binding MT3 (ML2) (agonist radioligand) 0088
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Other receptors      Nicotinic
binding new protocol N muscle-type (antagonist radioligand) Human 0936
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binding N muscle-type (antagonist radioligand) - custom offer 0111
inquire
specific discount
binding N neuronal alpha4beta2 (agonist radioligand) Human 3029
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binding N neuronal alpha4beta2 (agonist radioligand) - custom offer 0110
inquire
specific discount
binding new protocol N neuronal alpha 7 (antagonist radioligand) Human 3010
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Other receptors      Purinergic
binding P2X (agonist radioligand) 0127
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Other receptors      Serotonin
binding 5-HT3 (antagonist radioligand) Human 0411
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Other receptors      Sigma
binding new assay sigma (non-selective) (agonist radioligand) Human 3500
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binding sigma1 (agonist radioligand) - custom offer 0147
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specific discount
binding new protocol sigma1 (agonist radioligand) Human 0889
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binding new assay sigma2 (agonist radioligand) Human 3468
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Phosphodiesterases
binding rolipram (antagonist radioligand) 0379
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Serotonin
binding 5-HT transporter (antagonist radioligand) Human 0439
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binding 5-HT transporter (antagonist radioligand) - custom offer 0145
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specific discount
Transduction signal enzymes      Inositol phosphate
binding IP3 (agonist radioligand) 0083
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min 16 wells specific discount
Voltage-gated channels      Ca2+ channels
binding Ca2+- L (dihydropyridine site) (antagonist radioligand) 0161
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binding Ca2+- L (diltiazem site) (benzothiazepines) (antagonist radioligand) 0162
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binding Ca2+- L (verapamil site) (phenylalkylamine) (antagonist radioligand) 0163
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binding new protocol Ca2+- N (antagonist radioligand) 0164
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Voltage-gated channels      K+ channels
binding hERG (membrane preparation) (antagonist radioligand) Human 1868
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binding KATP (antagonist radioligand) 0165
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binding KV (antagonist radioligand) 0166
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binding SKCa (antagonist radioligand) 0167
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